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WorksheetsHabib Dad's review Q
Total questions: 19
Worksheet time: 12mins
The following rxn is catalyzed by
Type III deiodinase
Type II deiodinase
Type I deiodinase
WOTF statements about L-Thyroxine are correct?
one chiral center
negatively charged under physiological conditions
amphoteric compound
prohormone
What is the name of the following thyroid drug?
TSH
TRH
Levothyroxine
Liothyronine
PTU
WOTF statements about Liothyronin (T3) pKa 8.4 are correct?
Liothyronine has one chiral center. L isomer is the active isomer
L-Thyroxine (T4) has longer half-life than Liothyronine (T3)
Liothyronine is an active hormone
Liothyronine is an amphoteric compound
Liothyronine has a longer half-life (1 week) than L-thyroxineLiothyronine
WOTF is/are pro-hormone (T4)?
Which function does this molecule have? Methimazole
inhibits 5'-deiodinase enzyme
inhibits 5-deiodinase enzyme
inhibits TSH receptor
inhibits TRH receptor
inhibits thyroid peroxidase enzyme
Which function does this molecule have? Propylthiouracil
inhibits 5-deiodinase
inhibits 5'-deiodinase
inhibits thyroid peroxidase enzyme
inhibits TRH receptor
inhibits 2'-deiodinase enzyme
Which of the following compounds is/are active hormone (T3)?
What is the name of the following drug?
TSH
Levothyroxine
Liothyronine
TRH
PTU
ALL of the following are truuu about Estradiol EXCEPT:
Biosynthesis requires the key enzyme aromatase
exhibiting high potentcy when administered parentally
estradiol is a CHIRAL compound
steroid analog
exhibiting high potency when administered orally
What is the purpose of the ethinyl group at C-17? Ethinyl estradiol
Ethinyl is a chemically inert group and prevent metabolic oxidation of C17 hydroxy group
Ethinyl is a chemically inert group and prevent metabolic oxidation of C3 hydroxyl group
Ethinyl is a chemically inert group and prevent metabolic reduction of C17 hydroxyl group
Ethinyl is a chemically inert group and prevent metabolic oxidation of C17 alkyne group
Ethinyl is a chemically inert group and prevent glucuronide conjugation of C17 hydroxyl group
WOTF statements are truuu about Ethinyl estradiol and Mestranol?
Mestranol is 3-O-methyl ether of Ethinyl estradiol
Ethinyl estradiol undergoes extensive enterohepatic recycling
Ethinyl estradiol undergoes extensive first-pass metabolism
Mestranol is a prodrug of Ethinyl estradiol
Mestranol is a prodrug
The agonist potency of the exogenous estrogens
Estradiol > Estriol > Estrone
Estradiol > Estrone > Estriol
Estriol > Estradiol > Estrone
Estrone > Estradiol > Estriol
Estrone > Estriol > Estradiol
SATA: 7a-aminophenylthioandrost-dienedione
synthetic testosterone
aromatose inhibitior
CYP19 inhibitor
steroid analog
inhibits the conversion of testosterone to estrogens
SATA: Anastrozole
synthetic testosterone
triazole analog
aromatose inhibitor
inhibits the conversion of testosterone to estrogens
CYP19 inhibitor
SATA: Ethisterone
synthetic testosterone
synthetic progestin
aromatase inhibitor
15-fold more active than progesterone when administered orally
steroid analog
SATA: Norethindrone
acetylation of 17b-OH of Norethindrone enhances progestin activity
acetylation of 17b-OH of Norethindrone increases the duraction of action
Norethindrone is a synthetic progestin
Norethindrone is a steroid analog
Norethindrone is an aromatose inhibitor
SATA: Testosterone 17b-:
-propionate (less bulky)
-enanthate
-undecanote
-cyclopentylpropionate
-cypionate (bulky)
Testosterone is more active when administered parentally than orally
Testosterone 17b-propionate is avail for IM administration
Testosterone 17b-enanthate is a prodrug
Testosterone 17b-cypionate has a longer duration of action of 1-2 weeks
Testosterone 17b-enanthate has a longer duration of action of 2-4 weeks
SATA: Fluoxymestrone
synthetic testosterone
orally active
aromatase inhibitor
steroid analog
the presence of 17a alkyl group reduces susceptibility to hepatic oxidative metabolism
